英文名稱 | Raloxifene hydrochloride | Keoxifene hydrochloride | LY156758 | LY139481 hydrochloride |
---|---|
中文名稱 | 鹽酸雷洛昔芬 |
CAS號 | 82640-04-8 |
分子式 | C28H28ClNO4S |
分子量 | 510.04 |
外觀 | Light yellow to yellow powder |
儲存條件 | 4°C, sealed storage, away from moisture |
英文名稱 | Raloxifene hydrochloride | Keoxifene hydrochloride | LY156758 | LY139481 hydrochloride |
---|---|
中文名稱 | 鹽酸雷洛昔芬 |
CAS號 | 82640-04-8 |
分子式 | C28H28ClNO4S |
分子量 | 510.04 |
外觀 | Light yellow to yellow powder |
儲存條件 | 4°C, sealed storage, away from moisture |
Raloxifene (LY156758, Keoxifene) HCl is a selective and orally active estrogen receptor modulator (SERM), which inhibits human cytosolic aldehyde oxidase-catalyzed phthalazine oxidation activity with IC50 of 5.7 nM.
Potent inhibition of human liver aldehyde oxidase by raloxifene.
PMID: 14709625 DOI: 10.1124/dmd.32.1.89
PMID: 20958960 PMCID: PMC2978204 DOI: 10.1186/1471-2407-10-566