英文名稱 | Ketanserin tartrate | R41468 tartrate |
---|---|
中文名稱 | 酒石酸酮色林 | 酮舍林酒石酸鹽 |
CAS號 | 83846-83-7 |
分子式 | C26H28FN3O9 |
分子量 | 545.51 |
外觀 | White to off-white powder |
儲存條件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
英文名稱 | Ketanserin tartrate | R41468 tartrate |
---|---|
中文名稱 | 酒石酸酮色林 | 酮舍林酒石酸鹽 |
CAS號 | 83846-83-7 |
分子式 | C26H28FN3O9 |
分子量 | 545.51 |
外觀 | White to off-white powder |
儲存條件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
Ketanserin (R41468) tartrate is a selective 5-HT2 receptor antagonist. Ketanserin tartrate also blocks hERG current (IhERG) in a concentration-dependent manner (IC50=0.11 μM).
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