英文名稱 | Rimonabant | SR141716 |
---|---|
中文名稱 | 利莫那班 |
CAS號 | 168273-06-1 |
分子式 | C22H21Cl3N4O |
分子量 | 463.79 |
外觀 | White to off-white powder |
儲存條件 | 4°C, sealed storage, away from moisture |
英文名稱 | Rimonabant | SR141716 |
---|---|
中文名稱 | 利莫那班 |
CAS號 | 168273-06-1 |
分子式 | C22H21Cl3N4O |
分子量 | 463.79 |
外觀 | White to off-white powder |
儲存條件 | 4°C, sealed storage, away from moisture |
Rimonabant (SR141716) is a highly potent, brain penetrated and selective central cannabinoid receptor (CB1) antagonist with a Ki of 1.8 nM. Rimonabant (SR141716) also inhibits Mycobacterial membrane protein Large 3 (MMPL3).
Crystal Structures of Membrane Transporter MmpL3, an Anti-TB Drug Target.
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