英文名稱 | Sitagliptin phosphate | MK-0431 phosphate |
---|---|
中文名稱 | 磷酸西他列汀 |
CAS號 | 654671-78-0 |
分子式 | C16H15F6N5O·H3O4P |
分子量 | 505.31 | 407.32(free) |
外觀 | White to off-white powder |
儲存條件 | 4°C, sealed storage, away from moisture and light |
英文名稱 | Sitagliptin phosphate | MK-0431 phosphate |
---|---|
中文名稱 | 磷酸西他列汀 |
CAS號 | 654671-78-0 |
分子式 | C16H15F6N5O·H3O4P |
分子量 | 505.31 | 407.32(free) |
外觀 | White to off-white powder |
儲存條件 | 4°C, sealed storage, away from moisture and light |
Sitagliptin phosphate (MK-0431 phosphate) is a potent inhibitor of DPP4 with an IC50 of 19 nM in Caco-2 cell extracts.
PMID: 22186413 DOI: 10.1210/en.2011-1732
PMID: 18299314 DOI: 10.2337/db07-1639